3-(Aminomethyl)-1,3-dihydro-2,1-benzoxaborol-1-ol is used as a reactant in the preparation of (benzofuranyl-3-carbonyl)(pyrrolidin-3-yl)pyrazolecarboxamide derivatives with tuberculostatic activity.
參考文獻
Encinas, L., et al.: J. Med. Chem., 57, 1276 (2014);