Standards; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;
應用
(3R,8S,9S,12S)-Atazanavir is an impurity of Atazanavir (A790051); a novel azapeptide HIV protease inhibitor (PI) and antiviral agent.
參考文獻
Palella, F.J. Jr., et al.: N. Engl. J. Med., 338(13), 853 (1998); Nolan, D., et al.: Drugs, 63(23), 2555 (2003); Musial, B.L., et al.: Am. J. Health Syst. Pharm., 61, 1365 (2004); Wood, R., et al.: J. Acquir. Immune Defic. Syndr., 36, 684 (2004)