Building Blocks; Pharmaceutical/API Drug Impurities/Metabolites;
應用
7-Bromo-6-chloro-4(3H)-quinazolinone is an important intermediate in the manufacturing of the anticoccidial drug (coccidiostat) halofuginone (Tempostatin).
參考文獻
Trager, W., et al.: Science, 193, 673 (1976), Chien, P., et al.: J. Med. Chem., 13, 867 (1970), Zhu, S., et al.: Bioorg. Med. Chem. Lett., 16, 1854 (2006),